PDB Information

PDB4V3U
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Novel 2,4-Disubstituted Pyrimidines as Potent, Selective, and Cell-Permeable Inhibitors of Neuronal Nitric Oxide Synthase.
Mukherjee, P., Li, H., Sevrioukova, I., Chreifi, G., Martasek, P., Roman, L.J., Poulos, T.L., Silverman, R.B.
J.Med.Chem.
HeaderOxidoreductase
Released2014-10-20
Resolution2.300
CATH Insert Date04 Jan, 2015

PDB Images (17)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 05 Jan, 2015 Chopped
B 05 Jan, 2015 Chopped
C 05 Jan, 2015 Chopped
D 05 Jan, 2015 Chopped

CATH Domains (12)

Domain ID Date inserted into CATH Superfamily CATH Status
4v3uA01 30 Jan, 2017 3.90.340.10 Assigned
4v3uA02 30 Jan, 2017 3.90.440.10 Assigned
4v3uA03 30 Jan, 2017 3.90.1230.10 Assigned
4v3uB01 30 Jan, 2017 3.90.340.10 Assigned
4v3uB02 30 Jan, 2017 3.90.440.10 Assigned
4v3uB03 30 Jan, 2017 3.90.1230.10 Assigned
4v3uC01 30 Jan, 2017 3.90.340.10 Assigned
4v3uC02 30 Jan, 2017 3.90.440.10 Assigned
4v3uC03 30 Jan, 2017 3.90.1230.10 Assigned
4v3uD01 30 Jan, 2017 3.90.340.10 Assigned
4v3uD02 30 Jan, 2017 3.90.440.10 Assigned
4v3uD03 30 Jan, 2017 3.90.1230.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P29475 NOS1_HUMAN Homo sapiens Nitric oxide synthase, brain
P29475 NOS1_HUMAN Homo sapiens Nitric oxide synthase, brain
P29475 NOS1_HUMAN Homo sapiens Nitric oxide synthase, brain
P29475 NOS1_HUMAN Homo sapiens Nitric oxide synthase, brain