PDB Information

PDB4UZH
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Sar156497 an Exquisitely Selective Inhibitor of Aurora Kinases.
Carry, J.C., Clerc, F.F., Minoux, H., Schio, L., Mauger, J., Nair, A., Parmantier, E., Le Moigne, R., Delorme, C., Nicolas, J.P., Krick, A., Abecassis, P.Y., Crocq-Stuerga, V., Pouzieux, S., Delarbre, L., Maignan, S., Bertrand, T., Bjergarde, K., Ma, N., Lachaud, S., Guizani, H., Lebel, R., Doerflinger, G., Monget, S., Perron, S., Gasse, F., Angouillant-Boniface, O., Filoche-Romme, B.J., Murer, M., Gontier, S., Prevost, C., Monteiro, M.L., Combeau, C.
J.Med.Chem.
HeaderTransferase
Released2014-09-05
Resolution2.000
CATH Insert Date30 Nov, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 01 Dec, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4uzhA01 03 Dec, 2014 3.30.200.20 Assigned
4uzhA02 03 Dec, 2014 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O14965 AURKA_HUMAN Homo sapiens Aurora kinase A