PDB Information

PDB4UIZ
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
The Discovery of I-Brd9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition.
Theodoulou, N.H., Bamborough, P., Bannister, A.J., Becher, I., Bit, R.A., Che, K.H., Chung, C., Dittmann, A., Drewes, G., Drewry, D.H., Gordon, L., Grandi, P., Leveridge, M., Lindon, M., Michon, A., Molnar, J., Robson, S.C., Tomkinson, N.C.O., Kouzarides, T., Prinjha, R.K., Humphreys, P.G.
J.Med.Chem.
HeaderTranscription
Released2015-04-03
Resolution1.190
CATH Insert Date28 Jun, 2015

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4uizA01 15 Jul, 2015 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4