PDB Information

PDB4TMF
MethodX-RAY DIFFRACTION
Host OrganismPichia pastoris
Gene SourceHomo sapiens
Primary Citation
Cyclic adenosine 5'-diphosphate ribose analogs without a "southern" ribose inhibit ADP-ribosyl cyclase-hydrolase CD38.
Swarbrick, J.M., Graeff, R., Zhang, H., Thomas, M.P., Hao, Q., Potter, B.V.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2014-06-01
Resolution2.050
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4tmfA01 13 Jul, 2015 1.20.82.10 Assigned
4tmfA02 13 Jul, 2015 3.40.50.720 Assigned
4tmfB01 15 Jul, 2015 1.20.82.10 Assigned
4tmfB02 15 Jul, 2015 3.40.50.720 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P28907 CD38_HUMAN Homo sapiens ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
P28907 CD38_HUMAN Homo sapiens ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1