PDB 4rrv
PDB Information
| PDB | 4RRV |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | A small-molecule mimic of a peptide docking motif inhibits the protein kinase PDK1.
Proc.Natl.Acad.Sci.USA
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2014-11-06 |
| Resolution | 1.410 |
| CATH Insert Date | 28 Dec, 2014 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 29 Dec, 2014 | Chopped |
| B | 29 Dec, 2014 | Rejected |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4rrvA01 | 06 Jan, 2015 | 3.30.200.20 | Assigned |
| 4rrvA02 | 06 Jan, 2015 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q16513 | PKN2_HUMAN | Homo sapiens | Serine/threonine-protein kinase N2 |
| O15530 | PDPK1_HUMAN | Homo sapiens | 3-phosphoinositide-dependent protein kinase 1 |
