PDB Information

PDB4RQV
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
A small-molecule mimic of a peptide docking motif inhibits the protein kinase PDK1.
Rettenmaier, T.J., Sadowsky, J.D., Thomsen, N.D., Chen, S.C., Doak, A.K., Arkin, M.R., Wells, J.A.
Proc.Natl.Acad.Sci.USA
HeaderTransferase/Transferase Inhibitor
Released2014-11-05
Resolution1.500
CATH Insert Date28 Dec, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Dec, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4rqvA01 06 Jan, 2015 3.30.200.20 Assigned
4rqvA02 06 Jan, 2015 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O15530 PDPK1_HUMAN Homo sapiens 3-phosphoinositide-dependent protein kinase 1