PDB Information

PDB4RN2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Variable Active Site Loop Conformations Accommodate the Binding of Macrocyclic Largazole Analogues to HDAC8.
Decroos, C., Clausen, D.J., Haines, B.E., Wiest, O., Williams, R.M., Christianson, D.W.
Biochemistry
HeaderHydrolase/Hydrolase Inhibitor
Released2014-10-22
Resolution2.390
CATH Insert Date28 Jun, 2015

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4rn2A00 10 Jul, 2015 3.40.800.20 Assigned
4rn2B00 10 Jul, 2015 3.40.800.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9BY41 HDAC8_HUMAN Homo sapiens Histone deacetylase 8
Q9BY41 HDAC8_HUMAN Homo sapiens Histone deacetylase 8