PDB Information

PDB4R5V
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourcePlasmodium falciparum FcB1/Columbia
Primary Citation
Two-Pronged Attack: Dual Inhibition of Plasmodium falciparum M1 and M17 Metalloaminopeptidases by a Novel Series of Hydroxamic Acid-Based Inhibitors.
Mistry, S.N., Drinkwater, N., Ruggeri, C., Sivaraman, K.K., Loganathan, S., Fletcher, S., Drag, M., Paiardini, A., Avery, V.M., Scammells, P.J., McGowan, S.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2014-08-22
Resolution2.100
CATH Insert Date09 Nov, 2014

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 10 Nov, 2014 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
4r5vA01 13 Nov, 2014 2.60.40.1730 Assigned
4r5vA02 13 Nov, 2014 3.30.2010.30 Assigned
4r5vA03 13 Nov, 2014 1.10.390.10 Assigned
4r5vA04 13 Nov, 2014 2.60.40.1840 Assigned
4r5vA05 13 Nov, 2014 1.25.50.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O96935 AMP1_PLAFQ Plasmodium falciparum FcB1/Columbia M1 family aminopeptidase