PDB Information

PDB4QVX
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of a Potent and Selective BCL-XL Inhibitor with in Vivo Activity.
Tao, Z.F., Hasvold, L., Wang, L., Wang, X., Petros, A.M., Park, C.H., Boghaert, E.R., Catron, N.D., Chen, J., Colman, P.M., Czabotar, P.E., Deshayes, K., Fairbrother, W.J., Flygare, J.A., Hymowitz, S.G., Jin, S., Judge, R.A., Koehler, M.F., Kovar, P.J., Lessene, G., Mitten, M.J., Ndubaku, C.O., Nimmer, P., Purkey, H.E., Oleksijew, A., Phillips, D.C., Sleebs, B.E., Smith, B.J., Smith, M.L., Tahir, S.K., Watson, K.G., Xiao, Y., Xue, J., Zhang, H., Zobel, K., Rosenberg, S.H., Tse, C., Leverson, J.D., Elmore, S.W., Souers, A.J.
ACS MED.CHEM.LETT.
HeaderApoptosis/Inhibitor
Released2014-07-16
Resolution2.100
CATH Insert Date16 Aug, 2015

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 17 Aug, 2015 Chopped
B 17 Aug, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4qvxA00 24 Aug, 2015 1.10.437.10 Assigned
4qvxB00 19 Aug, 2015 1.10.437.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q07817 B2CL1_HUMAN Homo sapiens Bcl-2-like protein 1
Q07817 B2CL1_HUMAN Homo sapiens Bcl-2-like protein 1
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