PDB Information

PDB4QRC
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
DFG-out Mode of Inhibition by an Irreversible Type-1 Inhibitor Capable of Overcoming Gate-Keeper Mutations in FGF Receptors.
Huang, Z., Tan, L., Wang, H., Liu, Y., Blais, S., Deng, J., Neubert, T.A., Gray, N.S., Li, X., Mohammadi, M.
Acs Chem.Biol.
HeaderTransferase/Transferase Inhibitor
Released2014-06-30
Resolution1.900
CATH Insert Date09 Nov, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 10 Nov, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4qrcA01 13 Nov, 2014 3.30.200.20 Assigned
4qrcA02 13 Nov, 2014 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P22455 FGFR4_HUMAN Homo sapiens Fibroblast growth factor receptor 4