PDB Information

PDB4QQN
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of Potent and Selective Allosteric Inhibitors of Protein Arginine Methyltransferase 3 (PRMT3).
Kaniskan, H.U., Eram, M.S., Zhao, K., Szewczyk, M.M., Yang, X., Schmidt, K., Luo, X., Xiao, S., Dai, M., He, F., Zang, I., Lin, Y., Li, F., Dobrovetsky, E., Smil, D., Min, S.J., Lin-Jones, J., Schapira, M., Atadja, P., Li, E., Barsyte-Lovejoy, D., Arrowsmith, C.H., Brown, P.J., Liu, F., Yu, Z., Vedadi, M., Jin, J.
J. Med. Chem.
HeaderTransferase
Released2014-06-27
Resolution2.080
CATH Insert Date28 Sep, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Sep, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4qqnA01 07 Oct, 2014 3.40.50.150 Assigned
4qqnA02 07 Oct, 2014 2.70.160.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60678 ANM3_HUMAN Homo sapiens Protein arginine N-methyltransferase 3