PDB Information

PDB4QIA
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-activity relationships of imidazole-derived 2-[N-carbamoylmethyl-alkylamino]acetic acids, dual binders of human insulin-degrading enzyme.
Charton, J., Gauriot, M., Totobenazara, J., Hennuyer, N., Dumont, J., Bosc, D., Marechal, X., Elbakali, J., Herledan, A., Wen, X., Ronco, C., Gras-Masse, H., Heninot, A., Pottiez, V., Landry, V., Staels, B., Liang, W.G., Leroux, F., Tang, W.J., Deprez, B., Deprez-Poulain, R.
Eur.J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2014-05-30
Resolution3.200
CATH Insert Date28 Jun, 2015

PDB Images (11)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
4qiaA01 10 Jul, 2015 3.30.830.10 Assigned
4qiaA02 10 Jul, 2015 3.30.830.10 Assigned
4qiaA03 10 Jul, 2015 3.30.830.10 Assigned
4qiaA04 10 Jul, 2015 3.30.830.10 Assigned
4qiaB01 10 Jul, 2015 3.30.830.10 Assigned
4qiaB02 10 Jul, 2015 3.30.830.10 Assigned
4qiaB03 10 Jul, 2015 3.30.830.10 Assigned
4qiaB04 10 Jul, 2015 3.30.830.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P14735 IDE_HUMAN Homo sapiens Insulin-degrading enzyme
P14735 IDE_HUMAN Homo sapiens Insulin-degrading enzyme