PDB Information

PDB4PX5
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery and Structure Guided Optimization of Diarylmethanesulfonamide Disruptors of GK-GKRP Binding
Pennington, L.D., Bartberger, M.D., Croghan, M.D., Andrews, K.L., Ashton, K.S., Bourbeau, M.P., Chen, J., Chmait, S., Cupple, R., Fotsch, C.
To be Published
HeaderSugar Binding Protein/Inhibitor
Released2014-03-21
Resolution2.200
CATH Insert Date28 Jun, 2015

PDB Images (9)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
4px5A01 10 Jul, 2015 3.40.50.10490 Assigned
4px5A02 10 Jul, 2015 Holding pen
4px5A03 10 Jul, 2015 Holding pen
4px5B01 09 Jul, 2015 3.40.50.10490 Assigned
4px5B02 09 Jul, 2015 Holding pen
4px5B03 09 Jul, 2015 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein