PDB Information

PDB4PS3
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Structural Basis for Isoform Selectivity in a Class of Benzothiazole Inhibitors of Phosphoinositide 3-Kinase gamma.
Collier, P.N., Martinez-Botella, G., Cornebise, M., Cottrell, K.M., Doran, J.D., Griffith, J.P., Mahajan, S., Maltais, F., Moody, C.S., Huck, E.P., Wang, T., Aronov, A.M.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2014-03-06
Resolution2.900
CATH Insert Date18 May, 2014

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 19 May, 2014 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
4ps3A01 21 May, 2014 3.10.20.90 Assigned
4ps3A02 21 May, 2014 2.60.40.150 Assigned
4ps3A03 21 May, 2014 1.25.40.70 Assigned
4ps3A04 21 May, 2014 3.30.1010.10 Assigned
4ps3A05 21 May, 2014 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P48736 PK3CG_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform