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PDB Information

PDB4PP3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Methyl substitution of a rexinoid agonist improves potency and reveals site of lipid toxicity.
Atigadda, V.R., Xia, G., Desphande, A., Boerma, L.J., Lobo-Ruppert, S., Grubbs, C.J., Smith, C.D., Brouillette, W.J., Muccio, D.D.
J.Med.Chem.
HeaderTranscription
Released2014-02-26
Resolution2.000
CATH Insert Date29 Jun, 2014

PDB Images (4)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 30 Jun, 2014 Chopped
B 30 Jun, 2014 Rejected

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4pp3A00 03 Jul, 2014 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P19793 RXRA_HUMAN Homo sapiens Retinoic acid receptor RXR-alpha
Q15596 NCOA2_HUMAN Homo sapiens Nuclear receptor coactivator 2
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