PDB Information

PDB4PMP
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Maximizing diversity from a kinase screen: identification of novel and selective pan-Trk inhibitors for chronic pain.
Stachel, S.J., Sanders, J.M., Henze, D.A., Rudd, M.T., Su, H.P., Li, Y., Nanda, K.K., Egbertson, M.S., Manley, P.J., Jones, K.L., Brnardic, E.J., Green, A., Grobler, J.A., Hanney, B., Leitl, M., Lai, M.T., Munshi, V., Murphy, D., Rickert, K., Riley, D., Krasowska-Zoladek, A., Daley, C., Zuck, P., Kane, S.A., Bilodeau, M.T.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2014-05-22
Resolution1.800
CATH Insert Date29 Jun, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 30 Jun, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4pmpA01 02 Jul, 2014 3.30.200.20 Assigned
4pmpA02 02 Jul, 2014 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P04629 NTRK1_HUMAN Homo sapiens High affinity nerve growth factor receptor