PDB Information

PDB4PM0
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of 2-(Cyclopentylamino)thieno[3,2-d]pyrimidin-4(3H)-one Derivatives as a New Series of Potent Phosphodiesterase 7 Inhibitors.
Kawai, K., Endo, Y., Asano, T., Amano, S., Sawada, K., Ueo, N., Takahashi, N., Sonoda, Y., Nagai, M., Kamei, N., Nagata, N.
J.Med.Chem.
HeaderHydrolase
Released2014-05-20
Resolution2.100
CATH Insert Date21 Dec, 2014

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 22 Dec, 2014 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4pm0A00 28 Dec, 2014 1.10.1300.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q13946 PDE7A_HUMAN Homo sapiens High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A