PDB Information

PDB4PLB
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceStaphylococcus aureus
Primary Citation
Oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad spectrum antibacterial agents.
Singh, S.B., Kaelin, D.E., Wu, J., Miesel, L., Tan, C.M., Meinke, P.T., Olsen, D., Lagrutta, A., Bradley, P., Lu, J., Patel, S., Rickert, K.W., Smith, R.F., Soisson, S., Wei, C., Fukuda, H., Kishii, R., Takei, M., Fukuda, Y.
Acs Med.Chem.Lett.
HeaderIsomerase/Isomerase Inhibitor/Dna
Released2014-05-16
Resolution2.690
CATH Insert Date29 Jun, 2014

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
B 30 Jun, 2014 Chopped
D 30 Jun, 2014 Chopped
E 30 Jun, 2014 Rejected
F 30 Jun, 2014 Rejected

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4plbB01 03 Jul, 2014 Holding pen
4plbB02 03 Jul, 2014 Holding pen
4plbD01 02 Jul, 2014 Holding pen
4plbD02 02 Jul, 2014 Holding pen

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P0A0K8 GYRB_STAAU Staphylococcus aureus DNA gyrase subunit B
P20831 GYRA_STAAU Staphylococcus aureus DNA gyrase subunit A
P0A0K8 GYRB_STAAU Staphylococcus aureus DNA gyrase subunit B
P20831 GYRA_STAAU Staphylococcus aureus DNA gyrase subunit A