PDB 4pk5
PDB Information
| PDB | 4PK5 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Crystal Structures and Structure-Activity Relationships of Imidazothiazole Derivatives as IDO1 Inhibitors.
Acs Med.Chem.Lett.
|
| Header | Oxidoreductase/Oxidoreductase Inhibitor |
| Released | 2014-05-13 |
| Resolution | 2.790 |
| CATH Insert Date | 14 Sep, 2014 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 15 Sep, 2014 | Chopped |
| B | 15 Sep, 2014 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4pk5A01 | 16 Sep, 2014 | 1.20.58.480 | Assigned |
| 4pk5A02 | 16 Sep, 2014 | Holding pen | |
| 4pk5B01 | 16 Sep, 2014 | 1.20.58.480 | Assigned |
| 4pk5B02 | 16 Sep, 2014 | Holding pen |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P14902 | I23O1_HUMAN | Homo sapiens | Indoleamine 2,3-dioxygenase 1 |
| P14902 | I23O1_HUMAN | Homo sapiens | Indoleamine 2,3-dioxygenase 1 |
