PDB Information

PDB4PK5
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Crystal Structures and Structure-Activity Relationships of Imidazothiazole Derivatives as IDO1 Inhibitors.
Tojo, S., Kohno, T., Tanaka, T., Kamioka, S., Ota, Y., Ishii, T., Kamimoto, K., Asano, S., Isobe, Y.
Acs Med.Chem.Lett.
HeaderOxidoreductase/Oxidoreductase Inhibitor
Released2014-05-13
Resolution2.790
CATH Insert Date14 Sep, 2014

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 15 Sep, 2014 Chopped
B 15 Sep, 2014 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4pk5A01 16 Sep, 2014 1.20.58.480 Assigned
4pk5A02 16 Sep, 2014 Holding pen
4pk5B01 16 Sep, 2014 1.20.58.480 Assigned
4pk5B02 16 Sep, 2014 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P14902 I23O1_HUMAN Homo sapiens Indoleamine 2,3-dioxygenase 1
P14902 I23O1_HUMAN Homo sapiens Indoleamine 2,3-dioxygenase 1