PDB Information

PDB4P8O
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceStaphylococcus aureus
Primary Citation
Second-generation antibacterial benzimidazole ureas: discovery of a preclinical candidate with reduced metabolic liability.
Grillot, A.L., Tiran, A.L., Shannon, D., Krueger, E., Liao, Y., O'Dowd, H., Tang, Q., Ronkin, S., Wang, T., Waal, N., Li, P., Lauffer, D., Sizensky, E., Tanoury, J., Perola, E., Grossman, T.H., Doyle, T., Hanzelka, B., Jones, S., Dixit, V., Ewing, N., Liao, S., Boucher, B., Jacobs, M., Bennani, Y., Charifson, P.S.
J.Med.Chem.
HeaderIsomerase
Released2014-03-31
Resolution2.400
CATH Insert Date09 Nov, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 10 Nov, 2014 Chopped
B 10 Nov, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4p8oA00 12 Nov, 2014 3.30.565.10 Assigned
4p8oB00 13 Nov, 2014 3.30.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q6GKU0 GYRB_STAAR Staphylococcus aureus subsp. aureus MRSA252 DNA gyrase subunit B
Q6GKU0 GYRB_STAAR Staphylococcus aureus subsp. aureus MRSA252 DNA gyrase subunit B
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