PDB Information

PDB4P7E
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Triazolopyridines as Selective JAK1 Inhibitors: From Hit Identification to GLPG0634.
Menet, C.J., Fletcher, S.R., Van Lommen, G., Geney, R., Blanc, J., Smits, K., Jouannigot, N., Deprez, P., van der Aar, E.M., Clement-Lacroix, P., Lepescheux, L., Galien, R., Vayssiere, B., Nelles, L., Christophe, T., Brys, R., Uhring, M., Ciesielski, F., Van Rompaey, L.
J.Med.Chem.
HeaderTransferase
Released2014-03-27
Resolution2.400
CATH Insert Date30 Nov, 2014

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 01 Dec, 2014 Chopped
B 01 Dec, 2014 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4p7eA01 03 Dec, 2014 3.30.200.20 Assigned
4p7eA02 03 Dec, 2014 1.10.510.10 Assigned
4p7eB01 02 Dec, 2014 3.30.200.20 Assigned
4p7eB02 02 Dec, 2014 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O60674 JAK2_HUMAN Homo sapiens Tyrosine-protein kinase JAK2
O60674 JAK2_HUMAN Homo sapiens Tyrosine-protein kinase JAK2