PDB Information

PDB4OP2
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Small Molecule Disruptors of the Glucokinase-Glucokinase Regulatory Protein Interaction: 5. A Novel Aryl Sulfone Series, Optimization Through Conformational Analysis.
Tamayo, N.A., Norman, M.H., Bartberger, M.D., Hong, F.T., Bo, Y., Liu, L., Nishimura, N., Yang, K.C., Tadesse, S., Fotsch, C., Chen, J., Chmait, S., Cupples, R., Hale, C., Jordan, S.R., Lloyd, D.J., Sivits, G., Van, G., St Jean, D.J.
J.Med.Chem.
HeaderCarbohydrate Binding Protein/Inhibitor
Released2014-02-04
Resolution2.240
CATH Insert Date10 Aug, 2014

PDB Images (9)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 11 Aug, 2014 Chopped
B 11 Aug, 2014 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
4op2A01 20 Aug, 2014 3.40.50.10490 Assigned
4op2A02 20 Aug, 2014 Holding pen
4op2A03 20 Aug, 2014 Holding pen
4op2B01 20 Aug, 2014 3.40.50.10490 Assigned
4op2B02 20 Aug, 2014 Holding pen
4op2B03 20 Aug, 2014 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein