PDB Information

PDB4OGI
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Dual kinase-bromodomain inhibitors for rationally designed polypharmacology.
Ciceri, P., Muller, S., O'Mahony, A., Fedorov, O., Filippakopoulos, P., Hunt, J.P., Lasater, E.A., Pallares, G., Picaud, S., Wells, C., Martin, S., Wodicka, L.M., Shah, N.P., Treiber, D.K., Knapp, S.
Nat.Chem.Biol.
HeaderTranscription/Inhibitor
Released2014-01-16
Resolution1.730
CATH Insert Date09 Mar, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 10 Mar, 2014 Chopped
B 10 Mar, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4ogiA01 25 Apr, 2014 1.20.920.10 Assigned
4ogiB01 25 Apr, 2014 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4