PDB Information

PDB4OGB
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
The PDE inhibition profile of LY294002 and tetrahydropyranyl analogues reveals a chromone motif for the development of PDE inhibitors
Howard, B.L., Nankervis, J.L., Feil, S.C., Manallack, D.T., Holien, J.K., Zhen, Z., Jennings, I.G., Abbott, B.M., Parker, M.W., Thompson, P.E.
To be Published
HeaderHydrolase/Hydrolase Inhibitor
Released2014-01-15
Resolution2.030
CATH Insert Date28 Jun, 2015

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped
C 29 Jun, 2015 Chopped
D 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4ogbA00 09 Jul, 2015 1.10.1300.10 Assigned
4ogbB00 09 Jul, 2015 1.10.1300.10 Assigned
4ogbC00 10 Jul, 2015 1.10.1300.10 Assigned
4ogbD00 10 Jul, 2015 1.10.1300.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q08499 PDE4D_HUMAN Homo sapiens cAMP-specific 3',5'-cyclic phosphodiesterase 4D
Q08499 PDE4D_HUMAN Homo sapiens cAMP-specific 3',5'-cyclic phosphodiesterase 4D
Q08499 PDE4D_HUMAN Homo sapiens cAMP-specific 3',5'-cyclic phosphodiesterase 4D
Q08499 PDE4D_HUMAN Homo sapiens cAMP-specific 3',5'-cyclic phosphodiesterase 4D