PDB 4occ
PDB Information
PDB | 4OCC |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Novel Inhibitors of the MDM2-p53 Interaction Featuring Hydrogen Bond Acceptors as Carboxylic Acid Isosteres.
J.Med.Chem.
|
Header | Ligase/Ligase Inhibitor |
Released | 2014-01-08 |
Resolution | 1.800 |
CATH Insert Date | 06 Apr, 2014 |
PDB Images (7)
PDB Prints
PDB Chains (3)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 07 Apr, 2014 | Chopped |
C | 07 Apr, 2014 | Chopped |
E | 07 Apr, 2014 | Chopped |
CATH Domains (3)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4occA00 | 25 Apr, 2014 | 1.10.245.10 | Assigned |
4occC00 | 25 Apr, 2014 | 1.10.245.10 | Assigned |
4occE00 | 25 Apr, 2014 | 1.10.245.10 | Assigned |
UniProtKB Entries (3)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q00987 | MDM2_HUMAN | Homo sapiens | E3 ubiquitin-protein ligase Mdm2 |
Q00987 | MDM2_HUMAN | Homo sapiens | E3 ubiquitin-protein ligase Mdm2 |
Q00987 | MDM2_HUMAN | Homo sapiens | E3 ubiquitin-protein ligase Mdm2 |