PDB Information

PDB4OBE
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
In situ selectivity profiling and crystal structure of SML-8-73-1, an active site inhibitor of oncogenic K-Ras G12C.
Hunter, J.C., Gurbani, D., Ficarro, S.B., Carrasco, M.A., Lim, S.M., Choi, H.G., Xie, T., Marto, J.A., Chen, Z., Gray, N.S., Westover, K.D.
Proc.Natl.Acad.Sci.USA
HeaderHydrolase
Released2014-01-07
Resolution1.240
CATH Insert Date15 Jun, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Jun, 2014 Chopped
B 16 Jun, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4obeA00 18 Jun, 2014 3.40.50.300 Assigned
4obeB00 18 Jun, 2014 3.40.50.300 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P01116 RASK_HUMAN Homo sapiens GTPase KRas
P01116 RASK_HUMAN Homo sapiens GTPase KRas