PDB 4o97
PDB Information
| PDB | 4O97 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-guided discovery of 1,3,5 tri-substituted benzenes as potent and selective matriptase inhibitors exhibiting in vivo antitumor efficacy.
Bioorg.Med.Chem.
|
| Header | Hydrolase/Hydrolase Inhibitor |
| Released | 2014-01-02 |
| Resolution | 2.200 |
| CATH Insert Date | 01 Jun, 2014 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 02 Jun, 2014 | Chopped |
| B | 02 Jun, 2014 | Rejected |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4o97A01 | 03 Jun, 2014 | 2.40.10.10 | Assigned |
| 4o97A02 | 03 Jun, 2014 | 2.40.10.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9Y5Y6 | ST14_HUMAN | Homo sapiens | Suppressor of tumorigenicity 14 protein |
| Q9Y5Y6 | ST14_HUMAN | Homo sapiens | Suppressor of tumorigenicity 14 protein |
