PDB Information

PDB4NY9
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of the CCR1 antagonist, BMS-817399, for the treatment of rheumatoid arthritis.
Santella, J.B., Gardner, D.S., Duncia, J.V., Wu, H., Dhar, M., Cavallaro, C., Tebben, A.J., Carter, P.H., Barrish, J.C., Yarde, M., Briceno, S.W., Cvijic, M.E., Grafstrom, R.R., Liu, R., Patel, S.R., Watson, A.J., Yang, G., Rose, A.V., Vickery, R.D., Caceres-Cortes, J., Caporuscio, C., Camac, D.M., Khan, J.A., An, Y., Foster, W.R., Davies, P., Hynes, J.
J.Med.Chem.
HeaderTranscription/Transcription Inhibitor
Released2013-12-10
Resolution2.800
CATH Insert Date07 Sep, 2014

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Sep, 2014 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4ny9A00 10 Sep, 2014 1.10.565.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O75469 NR1I2_HUMAN Homo sapiens Nuclear receptor subfamily 1 group I member 2