PDB 4n4t
PDB Information
| PDB | 4N4T |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Mus musculus |
| Primary Citation | Structure-based design of 2-aminopyridine oxazolidinones as potent and selective tankyrase inhibitors.
ACS Med Chem Lett
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2013-10-08 |
| Resolution | 2.320 |
| CATH Insert Date | 15 Dec, 2013 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 16 Dec, 2013 | Chopped |
| B | 16 Dec, 2013 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4n4tA00 | 20 Dec, 2013 | 3.90.228.10 | Assigned |
| 4n4tB00 | 20 Dec, 2013 | 3.90.228.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q6PFX9 | TNKS1_MOUSE | Mus musculus | Poly [ADP-ribose] polymerase tankyrase-1 |
| Q6PFX9 | TNKS1_MOUSE | Mus musculus | Poly [ADP-ribose] polymerase tankyrase-1 |
