PDB Information

PDB4MZS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMus musculus
Primary Citation
Identification of potent and selective cathepsin S inhibitors containing different central cyclic scaffolds.
Hilpert, H., Mauser, H., Humm, R., Anselm, L., Kuehne, H., Hartmann, G., Gruener, S., Banner, D.W., Benz, J., Gsell, B., Kuglstatter, A., Stihle, M., Thoma, R., Sanchez, R.A., Iding, H., Wirz, B., Haap, W.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2013-09-30
Resolution1.850
CATH Insert Date24 Aug, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 25 Aug, 2014 Chopped
B 25 Aug, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4mzsA00 29 Aug, 2014 3.90.70.10 Assigned
4mzsB00 29 Aug, 2014 3.90.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O70370 CATS_MOUSE Mus musculus Cathepsin S
O70370 CATS_MOUSE Mus musculus Cathepsin S