PDB Information

PDB4MVH
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design, Optimization, and Biological Evaluation of Novel Keto-Benzimidazoles as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A).
Hu, E., Kunz, R.K., Chen, N., Rumfelt, S., Siegmund, A., Andrews, K., Chmait, S., Zhao, S., Davis, C., Chen, H., Lester-Zeiner, D., Ma, J., Biorn, C., Shi, J., Porter, A., Treanor, J., Allen, J.R.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2013-09-24
Resolution2.500
CATH Insert Date27 Oct, 2013

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 28 Oct, 2013 Chopped
B 28 Oct, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4mvhA00 02 Nov, 2013 1.10.1300.10 Assigned
4mvhB00 02 Nov, 2013 1.10.1300.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9Y233 PDE10_HUMAN Homo sapiens cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
Q9Y233 PDE10_HUMAN Homo sapiens cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A