PDB 4mqu

PDB Links
Overview

PDB Information

PDB	4MQU
Method	X-RAY DIFFRACTION
Host Organism	Spodoptera frugiperda
Gene Source	Homo sapiens
Primary Citation	Small molecule disruptors of the glucokinase-glucokinase regulatory protein interaction: 2. Leveraging structure-based drug design to identify analogues with improved pharmacokinetic profiles. St Jean, D.J., Ashton, K.S., Bartberger, M.D., Chen, J., Chmait, S., Cupples, R., Galbreath, E., Helmering, J., Hong, F.T., Jordan, S.R., Liu, L., Kunz, R.K., Michelsen, K., Nishimura, N., Pennington, L.D., Poon, S.F., Reid, D., Sivits, G., Stec, M.M., Tadesse, S., Tamayo, N., Van, G., Yang, K.C., Zhang, J., Norman, M.H., Fotsch, C., Lloyd, D.J., Hale, C. J.Med.Chem.
Header	Transferase Inhibitor
Released	2013-09-16
Resolution	2.220
CATH Insert Date	11 May, 2014

PDB Images (9)

Image of CATH 4mqu

4mqu

PDB 4mqu

Image of CATH 4mquA

4mquA

PDB Chain 4mquA

Image of CATH 4mquB

4mquB

PDB Chain 4mquB

Image of CATH 4mquA01

4mquA01

CATH Domain 4mquA01

Image of CATH 4mquA02

4mquA02

CATH Domain 4mquA02

Image of CATH 4mquA03

4mquA03

CATH Domain 4mquA03

Image of CATH 4mquB01

4mquB01

CATH Domain 4mquB01

Image of CATH 4mquB02

4mquB02

CATH Domain 4mquB02

Image of CATH 4mquB03

4mquB03

CATH Domain 4mquB03

PDB Prints

PDB Chains (2)

Chain ID	Date inserted into CATH	CATH Status
A	12 May, 2014	Chopped
B	12 May, 2014	Chopped

CATH Domains (6)

Domain ID	Date inserted into CATH	Superfamily	CATH Status
4mquA01	17 May, 2014	3.40.50.10490	Assigned
4mquA02	17 May, 2014		Holding pen
4mquA03	17 May, 2014		Holding pen
4mquB01	17 May, 2014	3.40.50.10490	Assigned
4mquB02	17 May, 2014		Holding pen
4mquB03	17 May, 2014		Holding pen

UniProtKB Entries (2)

Accession	Gene ID	Taxon	Description
Q14397	GCKR_HUMAN	Homo sapiens	Glucokinase regulatory protein
Q14397	GCKR_HUMAN	Homo sapiens	Glucokinase regulatory protein