PDB 4mpc
PDB Information
| PDB | 4MPC |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-guided Development of Specific Pyruvate Dehydrogenase Kinase Inhibitors Targeting the ATP-binding Pocket.
J.Biol.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2013-09-12 |
| Resolution | 1.700 |
| CATH Insert Date | 05 Jan, 2014 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 06 Jan, 2014 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4mpcA01 | 09 Jan, 2014 | 1.20.140.20 | Assigned |
| 4mpcA02 | 09 Jan, 2014 | 3.30.565.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q15119 | PDK2_HUMAN | Homo sapiens | [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial |
