PDB Information

PDB4MHA
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHomo sapiens
Primary Citation
Discovery of Mer specific tyrosine kinase inhibitors for the treatment and prevention of thrombosis.
Zhang, W., McIver, A.L., Stashko, M.A., DeRyckere, D., Branchford, B.R., Hunter, D., Kireev, D., Miley, M.J., Norris-Drouin, J., Stewart, W.M., Lee, M., Sather, S., Zhou, Y., Di Paola, J.A., Machius, M., Janzen, W.P., Earp, H.S., Graham, D.K., Frye, S.V., Wang, X.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2013-08-29
Resolution2.590
CATH Insert Date25 May, 2014

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 26 May, 2014 Chopped
B 26 May, 2014 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4mhaA01 28 May, 2014 3.30.200.20 Assigned
4mhaA02 28 May, 2014 1.10.510.10 Assigned
4mhaB01 28 May, 2014 3.30.200.20 Assigned
4mhaB02 28 May, 2014 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q12866 MERTK_HUMAN Homo sapiens Tyrosine-protein kinase Mer
Q12866 MERTK_HUMAN Homo sapiens Tyrosine-protein kinase Mer