PDB Information

PDB4MF3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
GluK1 antagonists from 6-(tetrazolyl)phenyl decahydroisoquinoline derivatives: in vitro profile and in vivo analgesic efficacy.
Martinez-Perez, J.A., Iyengar, S., Shannon, H.E., Bleakman, D., Alt, A., Clawson, D.K., Arnold, B.M., Bell, M.G., Bleisch, T.J., Castano, A.M., Del Prado, M., Dominguez, E., Escribano, A.M., Filla, S.A., Ho, K.H., Hudziak, K.J., Jones, C.K., Mateo, A., Mathes, B.M., Mattiuz, E.L., Ogden, A.M., Simmons, R.M., Stack, D.R., Stratford, R.E., Winter, M.A., Wu, Z., Ornstein, P.L.
Bioorg.Med.Chem.Lett.
HeaderSignaling Protein
Released2013-08-27
Resolution3.000
CATH Insert Date11 May, 2014

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 12 May, 2014 Chopped
B 12 May, 2014 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4mf3A01 17 May, 2014 3.40.190.10 Assigned
4mf3A02 17 May, 2014 3.40.190.10 Assigned
4mf3B01 17 May, 2014 3.40.190.10 Assigned
4mf3B02 17 May, 2014 3.40.190.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P39086 GRIK1_HUMAN Homo sapiens Glutamate receptor ionotropic, kainate 1
P39086 GRIK1_HUMAN Homo sapiens Glutamate receptor ionotropic, kainate 1