PDB 4m7b
PDB Information
| PDB | 4M7B |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Design, Synthesis, Crystallographic Studies, and Preliminary Biological Appraisal of New Substituted Triazolo[4,3-b]pyridazin-8-amine Derivatives as Tankyrase Inhibitors.
J.Med.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2013-08-12 |
| Resolution | 1.950 |
| CATH Insert Date | 16 Mar, 2014 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 17 Mar, 2014 | Chopped |
| C | 17 Mar, 2014 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4m7bA00 | 25 Apr, 2014 | 3.90.228.10 | Assigned |
| 4m7bC00 | 17 Apr, 2014 | 3.90.228.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9H2K2 | TNKS2_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-2 |
| Q9H2K2 | TNKS2_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-2 |
