PDB 4l32
PDB Information
| PDB | 4L32 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of tankyrase inhibiting flavones with increased potency and isoenzyme selectivity.
J.Med.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2013-06-05 |
| Resolution | 1.850 |
| CATH Insert Date | 03 Nov, 2013 |
PDB Images (9)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 04 Nov, 2013 | Chopped |
| B | 04 Nov, 2013 | Chopped |
| C | 04 Nov, 2013 | Chopped |
| D | 04 Nov, 2013 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4l32A00 | 08 Nov, 2013 | 3.90.228.10 | Assigned |
| 4l32B00 | 08 Nov, 2013 | 3.90.228.10 | Assigned |
| 4l32C00 | 08 Nov, 2013 | 6.20.320.10 | Assigned |
| 4l32D00 | 08 Nov, 2013 | 6.20.320.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9H2K2 | TNKS2_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-2 |
| Q9H2K2 | TNKS2_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-2 |
| Q9H2K2 | TNKS2_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-2 |
| Q9H2K2 | TNKS2_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase tankyrase-2 |
