PDB 4ksp
PDB Information
| PDB | 4KSP |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of a Selective Kinase Inhibitor (TAK-632) Targeting Pan-RAF Inhibition: Design, Synthesis, and Biological Evaluation of C-7-Substituted 1,3-Benzothiazole Derivatives.
J.Med.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2013-05-17 |
| Resolution | 2.930 |
| CATH Insert Date | 04 Aug, 2013 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 05 Aug, 2013 | Chopped |
| B | 05 Aug, 2013 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4kspA01 | 14 Aug, 2013 | 3.30.200.20 | Assigned |
| 4kspA02 | 14 Aug, 2013 | 1.10.510.10 | Assigned |
| 4kspB01 | 14 Aug, 2013 | 3.30.200.20 | Assigned |
| 4kspB02 | 14 Aug, 2013 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P15056 | BRAF_HUMAN | Homo sapiens | Serine/threonine-protein kinase B-raf |
| P15056 | BRAF_HUMAN | Homo sapiens | Serine/threonine-protein kinase B-raf |
