PDB 4ksp
PDB Information
| PDB | 4KSP | 
| Method | X-RAY DIFFRACTION | 
| Host Organism | Spodoptera frugiperda | 
| Gene Source | Homo sapiens | 
| Primary Citation | Discovery of a Selective Kinase Inhibitor (TAK-632) Targeting Pan-RAF Inhibition: Design, Synthesis, and Biological Evaluation of C-7-Substituted 1,3-Benzothiazole Derivatives. J.Med.Chem. | 
| Header | Transferase/Transferase Inhibitor | 
| Released | 2013-05-17 | 
| Resolution | 2.930 | 
| CATH Insert Date | 04 Aug, 2013 | 
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status | 
|---|---|---|
| A | 05 Aug, 2013 | Chopped | 
| B | 05 Aug, 2013 | Chopped | 
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status | 
|---|---|---|---|
| 4kspA01 | 14 Aug, 2013 | 3.30.200.20 | Assigned | 
| 4kspA02 | 14 Aug, 2013 | 1.10.510.10 | Assigned | 
| 4kspB01 | 14 Aug, 2013 | 3.30.200.20 | Assigned | 
| 4kspB02 | 14 Aug, 2013 | 1.10.510.10 | Assigned | 
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description | 
|---|---|---|---|
| P15056 | BRAF_HUMAN | Homo sapiens | Serine/threonine-protein kinase B-raf | 
| P15056 | BRAF_HUMAN | Homo sapiens | Serine/threonine-protein kinase B-raf | 
