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PDB Information

PDB4K8A
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Fragment-based discovery of focal adhesion kinase inhibitors.
Gradler, U., Bomke, J., Musil, D., Dresing, V., Lehmann, M., Holzemann, G., Greiner, H., Esdar, C., Krier, M., Heinrich, T.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2013-04-18
Resolution2.910
CATH Insert Date22 Sep, 2013

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 23 Sep, 2013 Chopped
B 23 Sep, 2013 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4k8aA01 25 Sep, 2013 3.30.200.20 Assigned
4k8aA02 25 Sep, 2013 1.10.510.10 Assigned
4k8aB01 25 Sep, 2013 3.30.200.20 Assigned
4k8aB02 25 Sep, 2013 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q05397 FAK1_HUMAN Homo sapiens Focal adhesion kinase 1
Q05397 FAK1_HUMAN Homo sapiens Focal adhesion kinase 1
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