PDB 4k77
PDB Information
| PDB | 4K77 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Design and evaluation of novel 8-oxo-pyridopyrimidine Jak1/2 inhibitors.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2013-04-16 |
| Resolution | 2.400 |
| CATH Insert Date | 06 Oct, 2013 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 07 Oct, 2013 | Chopped |
| B | 07 Oct, 2013 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4k77A01 | 10 Oct, 2013 | 3.30.200.20 | Assigned |
| 4k77A02 | 10 Oct, 2013 | 1.10.510.10 | Assigned |
| 4k77B01 | 10 Oct, 2013 | 3.30.200.20 | Assigned |
| 4k77B02 | 10 Oct, 2013 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P23458 | JAK1_HUMAN | Homo sapiens | Tyrosine-protein kinase JAK1 |
| P23458 | JAK1_HUMAN | Homo sapiens | Tyrosine-protein kinase JAK1 |
