PDB Information

PDB4K5Z
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of Potent, Selective Chymase Inhibitors via Fragment Linking Strategies.
Taylor, S.J., Padyana, A.K., Abeywardane, A., Liang, S., Hao, M.H., De Lombaert, S., Proudfoot, J., Farmer, B.S., Li, X., Collins, B., Martin, L., Albaugh, D.R., Hill-Drzewi, M., Pullen, S.S., Takahashi, H.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2013-04-15
Resolution1.800
CATH Insert Date07 Jul, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4k5zA01 09 Aug, 2013 2.40.10.10 Assigned
4k5zA02 09 Aug, 2013 2.40.10.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P23946 CMA1_HUMAN Homo sapiens Chymase