PDB Information

PDB4K5P
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourcePlasmodium falciparum FcB1/Columbia
Primary Citation
Synthesis and Structure-Activity Relationships of Phosphonic Arginine Mimetics as Inhibitors of the M1 and M17 Aminopeptidases from Plasmodium falciparum.
Kannan Sivaraman, K., Paiardini, A., Sienczyk, M., Ruggeri, C., Oellig, C.A., Dalton, J.P., Scammells, P.J., Drag, M., McGowan, S.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2013-04-15
Resolution1.850
CATH Insert Date07 Jul, 2013

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
4k5pA01 09 Aug, 2013 2.60.40.1730 Assigned
4k5pA02 09 Aug, 2013 3.30.2010.30 Assigned
4k5pA03 09 Aug, 2013 1.10.390.10 Assigned
4k5pA04 09 Aug, 2013 2.60.40.1840 Assigned
4k5pA05 09 Aug, 2013 1.25.50.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O96935 AMP1_PLAFQ Plasmodium falciparum FcB1/Columbia M1 family aminopeptidase