PDB 4k1b
PDB Information
| PDB | 4K1B |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of novel pyrazolo[1,5-a]pyrimidines as potent pan-Pim inhibitors by structure- and property-based drug design.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2013-04-04 |
| Resolution | 2.080 |
| CATH Insert Date | 07 Jul, 2013 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 Jul, 2013 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4k1bA01 | 09 Aug, 2013 | 3.30.200.20 | Assigned |
| 4k1bA02 | 09 Aug, 2013 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P11309 | PIM1_HUMAN | Homo sapiens | Serine/threonine-protein kinase pim-1 |
