PDB 4jzr
PDB Information
| PDB | 4JZR |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Novel complex crystal structure of prolyl hydroxylase domain-containing protein 2 (PHD2): 2,8-Diazaspiro[4.5]decan-1-ones as potent, orally bioavailable PHD2 inhibitors
Bioorg.Med.Chem.
|
| Header | Oxidoreductase |
| Released | 2013-04-03 |
| Resolution | 2.100 |
| CATH Insert Date | 03 Nov, 2013 |
PDB Images (3)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 04 Nov, 2013 | Chopped |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4jzrA00 | 06 Nov, 2013 | 2.60.120.620 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9GZT9 | EGLN1_HUMAN | Homo sapiens | Egl nine homolog 1 |
