PDB Information

PDB4JPA
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Hydantoin based inhibitors of MMP13--discovery of AZD6605.
De Savi, C., Waterson, D., Pape, A., Lamont, S., Hadley, E., Mills, M., Page, K.M., Bowyer, J., Maciewicz, R.A.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2013-03-19
Resolution2.000
CATH Insert Date09 Mar, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 10 Mar, 2014 Chopped
B 10 Mar, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4jpaA00 25 Apr, 2014 3.40.390.10 Assigned
4jpaB00 25 Apr, 2014 3.40.390.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P45452 MMP13_HUMAN Homo sapiens Collagenase 3
P45452 MMP13_HUMAN Homo sapiens Collagenase 3