PDB Information

PDB4JDS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
SETD7 in complex with inhibitor PF-5426 and S-adenosyl-methionine
Dong, A., Wu, H., Zeng, H., El Bakkouri, M., Barsyte, D., Vedadi, M., Tatlock, J., Owen, D., Bunnage, M., Bountra, C., Arrowsmith, C.H., Edwards, A.M., Brown, P.J.
to be published
HeaderTransferase/Transferase Inhibitor
Released2013-02-25
Resolution1.700
CATH Insert Date07 Jul, 2013

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped
B 08 Jul, 2013 Chopped
C 08 Jul, 2013 Chopped
D 08 Jul, 2013 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
4jdsA01 09 Aug, 2013 2.20.110.10 Assigned
4jdsA02 09 Aug, 2013 2.170.270.10 Assigned
4jdsB01 09 Aug, 2013 2.20.110.10 Assigned
4jdsB02 09 Aug, 2013 2.170.270.10 Assigned
4jdsC01 09 Aug, 2013 2.20.110.10 Assigned
4jdsC02 09 Aug, 2013 2.170.270.10 Assigned
4jdsD01 09 Aug, 2013 2.20.110.10 Assigned
4jdsD02 09 Aug, 2013 2.170.270.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q8WTS6 SETD7_HUMAN Homo sapiens Histone-lysine N-methyltransferase SETD7
Q8WTS6 SETD7_HUMAN Homo sapiens Histone-lysine N-methyltransferase SETD7
Q8WTS6 SETD7_HUMAN Homo sapiens Histone-lysine N-methyltransferase SETD7
Q8WTS6 SETD7_HUMAN Homo sapiens Histone-lysine N-methyltransferase SETD7