PDB Information

PDB4JAJ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
SAR and evaluation of novel 5H-benzo[c][1,8]naphthyridin-6-one analogs as Aurora kinase inhibitors.
Karra, S., Xiao, Y., Chen, X., Liu-Bujalski, L., Huck, B., Sutton, A., Goutopoulos, A., Askew, B., Josephson, K., Jiang, X., Shutes, A., Shankar, V., Noonan, T., Garcia-Berrios, G., Dong, R., Dhanabal, M., Tian, H., Wang, Z., Clark, A., Goodstal, S.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2013-02-18
Resolution2.700
CATH Insert Date07 Jul, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4jajA01 09 Aug, 2013 3.30.200.20 Assigned
4jajA02 09 Aug, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O14965 AURKA_HUMAN Homo sapiens Aurora kinase A