PDB Information

PDB4J3F
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceFrancisella tularensis subsp. tularensis
Primary Citation
Structural and biological evaluation of a novel series of benzimidazole inhibitors of Francisella tularensis enoyl-ACP reductase (FabI).
Mehboob, S., Song, J., Hevener, K.E., Su, P.C., Boci, T., Brubaker, L., Truong, L., Mistry, T., Deng, J., Cook, J.L., Santarsiero, B.D., Ghosh, A.K., Johnson, M.E.
Bioorg.Med.Chem.Lett.
HeaderOxidoreductase/Oxidoreductase Inhibitor
Released2013-02-05
Resolution1.850
CATH Insert Date10 Aug, 2014

PDB Images (17)

PDB Prints

PDB Chains (8)

Chain ID Date inserted into CATH CATH Status
A 11 Aug, 2014 Chopped
B 11 Aug, 2014 Chopped
C 11 Aug, 2014 Chopped
D 11 Aug, 2014 Chopped
E 11 Aug, 2014 Chopped
F 11 Aug, 2014 Chopped
G 11 Aug, 2014 Chopped
H 11 Aug, 2014 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
4j3fA00 20 Aug, 2014 3.40.50.720 Assigned
4j3fB00 20 Aug, 2014 3.40.50.720 Assigned
4j3fC00 20 Aug, 2014 3.40.50.720 Assigned
4j3fD00 20 Aug, 2014 3.40.50.720 Assigned
4j3fE00 20 Aug, 2014 3.40.50.720 Assigned
4j3fF00 20 Aug, 2014 3.40.50.720 Assigned
4j3fG00 20 Aug, 2014 3.40.50.720 Assigned
4j3fH00 20 Aug, 2014 3.40.50.720 Assigned

UniProtKB Entries (8)

Accession Gene ID Taxon Description
Q5NGQ3 Q5NGQ3_FRATT Francisella tularensis subsp. tularensis SCHU S4 Enoyl-[acyl-carrier-protein] reductase [NADH]
Q5NGQ3 Q5NGQ3_FRATT Francisella tularensis subsp. tularensis SCHU S4 Enoyl-[acyl-carrier-protein] reductase [NADH]
Q5NGQ3 Q5NGQ3_FRATT Francisella tularensis subsp. tularensis SCHU S4 Enoyl-[acyl-carrier-protein] reductase [NADH]
Q5NGQ3 Q5NGQ3_FRATT Francisella tularensis subsp. tularensis SCHU S4 Enoyl-[acyl-carrier-protein] reductase [NADH]
Q5NGQ3 Q5NGQ3_FRATT Francisella tularensis subsp. tularensis SCHU S4 Enoyl-[acyl-carrier-protein] reductase [NADH]
Q5NGQ3 Q5NGQ3_FRATT Francisella tularensis subsp. tularensis SCHU S4 Enoyl-[acyl-carrier-protein] reductase [NADH]
Q5NGQ3 Q5NGQ3_FRATT Francisella tularensis subsp. tularensis SCHU S4 Enoyl-[acyl-carrier-protein] reductase [NADH]
Q5NGQ3 Q5NGQ3_FRATT Francisella tularensis subsp. tularensis SCHU S4 Enoyl-[acyl-carrier-protein] reductase [NADH]