PDB Information

PDB4J3E
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceXenopus laevis
Primary Citation
Discovery of RG7112: A Small-Molecule MDM2 Inhibitor in Clinical Development.
Vu, B., Wovkulich, P., Pizzolato, G., Lovey, A., Ding, Q., Jiang, N., Liu, J.J., Zhao, C., Glenn, K., Wen, Y., Tovar, C., Packman, K., Vassilev, L., Graves, B.
ACS Med Chem Lett
HeaderLigase/Antagonist
Released2013-02-05
Resolution1.910
CATH Insert Date07 Jul, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4j3eA00 09 Aug, 2013 1.10.245.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P56273 MDM2_XENLA Xenopus laevis E3 ubiquitin-protein ligase Mdm2