PDB Information

PDB4J1R
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Fragment-based approach using diversity-oriented synthesis yields a GSK3b inhibitor
Wang, Y., Wach, J., Sheehan, P., Zhong, C., Zhan, C., Harris, R., Almo, S.C., Bishop, J., Haggarty, S., Ramek, A., Berry, K., O'Herin, C., Koehler, A.N., Hung, A.W., Young, D.W.
To be Published
HeaderTransferase
Released2013-02-01
Resolution2.700
CATH Insert Date28 Mar, 2013

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 28 Mar, 2013 Chopped
B 28 Mar, 2013 Chopped
C 28 Mar, 2013 Chopped
D 28 Mar, 2013 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
4j1rA01 10 Apr, 2013 3.30.200.20 Assigned
4j1rA02 10 Apr, 2013 1.10.510.10 Assigned
4j1rB01 10 Apr, 2013 3.30.200.20 Assigned
4j1rB02 10 Apr, 2013 1.10.510.10 Assigned
4j1rC01 10 Apr, 2013 3.30.200.20 Assigned
4j1rC02 10 Apr, 2013 1.10.510.10 Assigned
4j1rD01 10 Apr, 2013 3.30.200.20 Assigned
4j1rD02 10 Apr, 2013 1.10.510.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P49841 GSK3B_HUMAN Homo sapiens Glycogen synthase kinase-3 beta
P49841 GSK3B_HUMAN Homo sapiens Glycogen synthase kinase-3 beta
P49841 GSK3B_HUMAN Homo sapiens Glycogen synthase kinase-3 beta
P49841 GSK3B_HUMAN Homo sapiens Glycogen synthase kinase-3 beta